Browsing by Subject "benzenesulfonamide derivative"

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Investigation on biological activities of anthranilic acid sulfonamide analogs

Doungsoongnuen S.; Worachartcheewan A.; Pingaew R.; Suksrichavalit T.; Prachayasittikul S.; Ruchirawat S.; Prachayasittikul V. (2011)

In the previous studies, the cytotoxicities of anthranilate sulfonamides were investigated. Herein, the bioactivities of 4-substituted (X = NO2, OCH3, CH3, Cl) benzenesulfonamides of anthranilic acid (5-8) are reported. ...
Synthesis and cytotoxicity of novel 4-(4-(substituted)-1H-1,2,3-triazol-1- yl)-N-phenethylbenzenesulfonamides

Pingaew R.; Prachayasittikul S.; Ruchirawat S.; Prachayasittikul V. (2014)

A new series of 4-(4-(substituted)-1H-1,2,3-triazol-1-yl)-N- phenethylbenzenesulfonamide derivatives 5 were synthesized through the Click approach and evaluated for their cytotoxic activity against four cancer cell lines ...
Synthesis, molecular docking, and QSAR study of bis-sulfonamide derivatives as potential aromatase inhibitors

Leechaisit R.; Pingaew R.; Prachayasittikul V.; Worachartcheewan A.; Prachayasittikul S.; Ruchirawat S.; Prachayasittikul V. (2019)

A library of bis-sulfonamides (9–26) were synthesized and tested for their aromatase inhibitory activities. Interestingly, all bis-sulfonamide derivatives inhibited the aromatase with IC50 range of 0.05–11.6 μM except for ...

Now showing items 1-3 of 3

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